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Synthesis and biological evaluation of 1,4-benzodiazepin-2-ones with antitrypanosomal activity

Synthesis and biological evaluation of 1,4-benzodiazepin-2-ones with antitrypanosomal activity,10.1016/j.bmc.2011.01.010,Bioorganic & Medicinal Chemis

Synthesis and biological evaluation of 1,4-benzodiazepin-2-ones with antitrypanosomal activity  
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A library of 1,4-benzodiazepines has been synthesized and evaluated against Trypanosoma brucei, a causative parasite of Human African trypanosomiasis. Benzodiazepines possessing a P2- transporter motif were found to have MIC values as low as 0.78μM.
Journal: Bioorganic & Medicinal Chemistry - BIOORGAN MED CHEM , vol. 19, no. 5, pp. 1802-1815, 2011
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